2-[[4-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-1H-吡唑-1-基]甲基]-吡啶合成路线 (共 1 条)
反应条件
1: 2-(1H-Pyrazole-4-yl)-4,4,5,5-tetramethyl-1,3,2-dioxaborolane With sodium hydride in N,N-dimethyl-formamide 0.5 h; 2: 2-chloromethyl-pyridine hydrochloride With tetra-(n-butyl)ammonium iodide
参考文献
US2011/281842 A1, ;
Page/Page column 59-60 ;