5-溴-2-环丙基异吲哚啉-1-酮合成路线 (共 2 条)
反应条件
potassium carbonate in ethanol
T=40°C; 3 h;
参考文献
INCYTE CORPORATION; ZHANG, Colin; QIAN, Ding-quan; ZHUO, Jincong; YAO, Wenqing
Patent: WO2010/75270 A1, 2010 ;
Location in patent: Page/Page column 184 ;
WO 2010/075270 A1
反应条件
triethylamine in toluene
Heating / reflux;
参考文献
BANYU PHARMACEUTICAL CO., LTD.
Patent: EP1726585 A1, 2006 ;
Location in patent: Page/Page column 48 ;