反应条件
1: 40.21 percent / 1.) sodium hydride / dimethylformamide / 1.) 0 deg C to 5 deg C, 2.) room temperature, 3 h
2: 57.1 percent / 3 h / 125 °C
View Scheme
参考文献
Pudlo, Jeffrey S.; Saxena, Naveen K.; Nassiri, M. Reza; Turk, Steven R.; Drach, John C.; Townsend, Leroy B.
Journal of Medicinal Chemistry, 1988 , vol. 31, # 11 p. 2086 - 2092