反应条件
1: 70 percent / POCl3, N,N-diethylaniline / 2 h / Heating
2: 45 percent / Na2CO3 / acetonitrile / 18 h / Heating
3: 80 percent / 30percent aq. H2O2, Na2WO4 / acetic acid / 16 h / 20 °C
View Scheme
参考文献
d'Atri; Gomarasca; Resnati; Tronconi; Scolastico; Sirtori
Journal of Medicinal Chemistry, 1984 , vol. 27, # 12 p. 1621 - 1629