反应条件
1: 83 percent / POCl3, N,N-diethylaniline / 13 h / 107 °C
2: 51.5 percent / NaOH / ethanol / 4 h / Heating
3: 80 percent / 30percent aq. NaOH / ethanol / 0.03 h / Heating
4: 32 percent / ethanol / 7 h / Heating
View Scheme
参考文献
d'Atri; Gomarasca; Resnati; Tronconi; Scolastico; Sirtori
Journal of Medicinal Chemistry, 1984 , vol. 27, # 12 p. 1621 - 1629