5-[(二甲基氨基)甲基]-2-甲酸合成路线 (共 1 条)
反应条件
1: dimethyl amine With sodium hydride in N,N-dimethyl-formamide T=20°C; 0.5 h; 2: 5-Chloromethyl-furan-2-carboxylic acid ethyl ester in N,N-dimethyl-formamide 48 h; 3: With sodium hydroxide; water in ethanol T=80°C; 0.666667 h;
参考文献
WO2005/89771 A1, ;
Page/Page column 38 ;
WO 2005/089771 A1