(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯合成路线

参考文献

Chu, Wenhua; Zhang, Jun; Zeng, Chenbo; Rothfuss, Justin; Tu, Zhude; Chu, Yunxiang; Reichert, David E.; Welch, Michael J.; Mach, Robert H.
Journal of Medicinal Chemistry, 2005 , vol. 48, # 24 p. 7637 - 7647

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

239483-09-1(S)-2-(氨乙基)-1-N-BOC-吡咯烷

参考文献

Comess, Kenneth M.; Erickson, Scott A.; Henkin, Jack; Kalvin, Douglas M.; Kawai, Megumi; Kim, Ki H.; BaMaung, Nwe Y.; Park, Chang Hoon; Sheppard, George S.; Vasudevan, Anil; Wang, Jieyi; Barnes, David M.; Fidanze, Steve D.; Kolaczkowski, Lawrence; Mantei, Robert A.; Park, David C.; Sanders, William J.; Tedrow, Jason S.; Wang, Gary T.
Patent: US2004/167128 A1, 2004 ;
Location in patent: Page 103 ;

69610-40-8N-Boc-L-脯氨醇+

104-15-4对甲苯磺酸

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

Dainippon Sumitomo Pharma Co., Ltd.; MARUYAMA, Megumi; KINOMURA, Naoya; NOJIMA, Satoshi; TAKAMURA, Masahiro; KAKIGUCHI, Keisuke; TATAMITANI, Hiroto
Patent: WO2011/111875 A1, 2011 ;
Location in patent: Page/Page column 64 ;
WO 2011/111875 A1

69610-40-8N-Boc-L-脯氨醇+

98-59-9对甲苯磺酰氯

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

Washington University in St. Louis
Patent: US2009/68105 A1, 2009 ;
Location in patent: Page/Page column 9 ;

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

SmithKline Beecham Corporation
Patent: US6514992 B1, 2003 ;
US 6514992 B1

24424-99-5二碳酸二叔丁酯

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

Alza, Esther; Cambeiro, Xacobe C.; Jimenez, Ciril; Pericas, Miquel A.
Organic Letters, 2007 , vol. 9, # 19 p. 3717 - 3720

23356-96-9L-脯氨醇

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

Alza, Esther; Cambeiro, Xacobe C.; Jimenez, Ciril; Pericas, Miquel A.
Organic Letters, 2007 , vol. 9, # 19 p. 3717 - 3720

147-85-3L-脯氨酸

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

Alza, Esther; Cambeiro, Xacobe C.; Jimenez, Ciril; Pericas, Miquel A.
Organic Letters, 2007 , vol. 9, # 19 p. 3717 - 3720

15761-39-4BOC-L-脯氨酸

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

Bartoli, Giuseppe; Bosco, Marcella; Dalpozzo, Renato; Giuliani, Arianna; Marcantoni, Enrico; Mecozzi, Tiziana; Sambri, Letizia; Torregiani, Elisabetta
Journal of Organic Chemistry, 2002 , vol. 67, # 25 p. 9111 - 9114

59936-29-7Boc-L-脯氨酸甲酯

86661-32-7(S)-2-(甲苯磺酰氧基甲基)吡咯烷-1-甲酸叔丁酯

参考文献

Cran; Gibson; Handa
Tetrahedron Asymmetry, 1995 , vol. 6, # 7 p. 1553 - 1556