6-氯-2-氟-3-甲氧基苯硼酸合成路线 (共 1 条)
反应条件
1: With n-butyllithium in tetrahydrofuran T=-78°C; 0.333333 h; 2: With boric acid trimethyl ester in tetrahydrofuran T=-78 - 20°C; 2 h; 3: With hydrogenchloride; water in tetrahydrofuran
参考文献
TargeGen, Inc.
Patent: US2005/245524 A1, 2005 ;
Location in patent: Page/Page column 97 ;
US 20050245524 A1