1: With diisobutylaluminium hydride in tetrahydrofuran; dichloromethane T=-78°C; 3 h; 2: With hydrogenchloride in tetrahydrofuran; dichloromethane; water
参考文献
MERCK and CO., INC.
Patent: WO2005/100356 A1, 2005 ;
Location in patent: Page/Page column 53-54 ;
WO 2005/100356 A1