反应条件
sodium hydride
1.) DMF, 0 deg C, 15 min, 2.) DMF, from 0 deg C to RT 3 h; Yield given. Multistep reaction;
参考文献
McKittrick, Brian A.; Ma, Ke; Huie, Keith; Yumibe, Nathan; Davis Jr., Harry; Clader, John W.; Czarniecki, Michael; McPhail, Andrew T.
Journal of Medicinal Chemistry, 1998 , vol. 41, # 5 p. 752 - 759