4-(4-氟-1H-吡咯并[2,3-B]吡啶-3-基)-2-噻唑胺合成路线 (共 1 条)
反应条件
1: in ethanol
T=70°C; 1 h;
2: With sodium carbonate in water
pH=~ 7.5;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2005/103050 A2, 2005 ;
Location in patent: Page/Page column 179-180 ;
WO 2005/103050 A2