1-丙酰基-2,3-二氢-1H-吲哚-5-磺酰氯合成路线 (共 2 条)
反应条件
1: pyridine / N,N-dimethyl-formamide / 0 - 20 °C
2: chlorosulfonic acid; phosphorus pentachloride / 0 - 80 °C
View Scheme
参考文献
Khan, Pasha M.; Correa, Ricardo G.; Divlianska, Daniela B.; Peddibhotla, Satyamaheshwar; Sessions, E. Hampton; Magnuson, Gavin; Brown, Brock; Suyama, Eigo; Yuan, Hongbin; Mangravita-Novo, Arianna; Vicchiarelli, Michael; Su, Ying; Vasile, Stefan; Smith, Layton H.; Diaz, Paul W.; Reed, John C.; Roth, Gregory P.
ACS Medicinal Chemistry Letters, 2011 , vol. 2, # 10 p. 780 - 785
反应条件
chlorosulfonic acid; phosphorus pentachloride
T=0 - 80°C;
参考文献
Khan, Pasha M.; Correa, Ricardo G.; Divlianska, Daniela B.; Peddibhotla, Satyamaheshwar; Sessions, E. Hampton; Magnuson, Gavin; Brown, Brock; Suyama, Eigo; Yuan, Hongbin; Mangravita-Novo, Arianna; Vicchiarelli, Michael; Su, Ying; Vasile, Stefan; Smith, Layton H.; Diaz, Paul W.; Reed, John C.; Roth, Gregory P.
ACS Medicinal Chemistry Letters, 2011 , vol. 2, # 10 p. 780 - 785