N-[2-(氨基甲基)苯基]-n-甲基甲烷磺酰胺合成路线 (共 1 条)
反应条件
1: caesium carbonate / N,N-dimethyl-formamide / 48 h / 20 °C
2: ammonia; methanol / Ra-Ni / 4 h / 20 °C / 1551.49 Torr
View Scheme
参考文献
ABBOTT LABORATORIES; ABBOTT LABORATORIES TRADING (SHANGHAI) COMPANY, LTD.; VAN CAMP, Jennifer; XU, Xiangdong; OSUMA, Augustine, Toby; GREGG, Robert; LONGENECKER, Kenton, L.
Patent: WO2012/45195 A1, 2012 ;
WO 2012/045195 A1