1: With tris-(dibenzylideneacetone)dipalladium(0); triphenylphosphine on polystyrene in tetrahydrofuran T=20°C; 0.25 h; 2: With triethylamine in tetrahydrofuran T=50°C; 1 h;
参考文献
NOVARTIS AG; NOVARTIS PHARMA GMBH
Patent: WO2007/147659 A1, 2007 ;
Location in patent: Page/Page column 30 ;
WO 2007/147659 A1
Angeles Castro; Miguel Del Corral, Jose M.; Garcia, Pablo A.; Victoria Rojo; Bento, Ana C.; Mollinedo, Faustino; Francesch, Andres M.; San Feliciano, Arturo
European Journal of Medicinal Chemistry, 2012 , vol. 58, p. 377 - 389