1-Boc-4-氨基哌啶合成路线

参考文献

Buckley, George M.; Ceska, Thomas A.; Fraser, Joanne L.; Gowers, Lewis; Groom, Colin R.; Higueruelo, Alicia Perez; Jenkins, Kerry; Mack, Stephen R.; Morgan, Trevor; Parry, David M.; Pitt, William R.; Rausch, Oliver; Richard, Marianna D.; Sabin, Verity
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87120-72-71-Boc-4-氨基哌啶

309251-30-7

参考文献

Huang; Hammond; Wu; Mach
Journal of Medicinal Chemistry, 2001 , vol. 44, # 25 p. 4404 - 4415

3132-99-8间溴苯甲醛+

87120-72-71-Boc-4-氨基哌啶

359877-98-84-[(3-溴苄基)氨基]-1-哌啶羧酸叔丁酯

参考文献

Seifert, Katrin; Buettner, Anita; Rigol, Stephan; Eilert, Nicole; Giannis, Athanassios; Wandel, Elke
Bioorganic and Medicinal Chemistry, 2012 , vol. 20, # 21 p. 6465 - 6481,17

87120-72-71-Boc-4-氨基哌啶+

350-46-9对氟硝基苯

333986-61-1

参考文献

Noguchi, Tetsuji; Tanaka, Naoki; Nishimata, Toyoki; Goto, Riki; Hayakawa, Miho; Sugidachi, Atsuhiro; Ogawa, Taketoshi; Asai, Fumitoshi; Ozeki, Tomoko; Fujimoto, Koichi
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1009-35-43-硝基-4-氟苯腈+

87120-72-71-Boc-4-氨基哌啶

320406-05-1

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PFIZER PRODUCTS INC.
Patent: WO2008/84300 A1, 2008 ;
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WO 2008/084300 A1

32315-10-9三光气+

87120-72-71-Boc-4-氨基哌啶

320581-97-32-甲基-2-丙基4-异氰酸-1-哌啶羧酸酯

参考文献

Zhang, Yongda; Li, Ning; Qu, Bo; Ma, Shengli; Lee, Heewon; Gonnella, Nina C.; Gao, Joe; Li, Wenjie; Tan, Zhulin; Reeves, Jonathan T.; Wang, Jun; Lorenz, Jon C.; Li, Guisheng; Reeves, Diana C.; Premasiri, Ajith; Grinberg, Nelu; Haddad, Nizar; Lu, Bruce Z.; Song, Jinhua J.; Senanayake, Chris H.
Organic Letters, 2013 , vol. 15, # 7 p. 1710 - 1713

75-44-5光气+

87120-72-71-Boc-4-氨基哌啶

320581-97-32-甲基-2-丙基4-异氰酸-1-哌啶羧酸酯

参考文献

Chaturvedula, Prasad V.; Mercer, Stephen E.; Fang, Haiquan
Patent: US2006/94707 A1, 2006 ;
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US 20060094707 A1

87120-72-71-Boc-4-氨基哌啶

125541-22-21-N-Boc-4-苯胺基哌啶

参考文献

Bioorganic and Medicinal Chemistry Letters, , vol. 13, # 3 p. 427 - 431

87120-72-71-Boc-4-氨基哌啶+

75-07-0乙醛

264905-39-71-N-Boc-4-乙胺哌啶

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SANOFI-AVENTIS
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Location in patent: Page/Page column 57-58 ;
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87120-72-71-Boc-4-氨基哌啶+

501-53-1氯甲酸苄酯

220394-97-81-Boc-4-Cbz-氨基哌啶