4-乙氧基3-三氟甲基苯硼酸合成路线 (共 1 条)
反应条件
1: With n-butyllithium in tetrahydrofuran; hexanes; water T=-78 - -70°C; 0.0833333 h; 2: With tri-isopropoxy-borane in tetrahydrofuran; hexanes T=-78°C; 0.5 h; 3: With acetic acid in tetrahydrofuran; hexanes; water
参考文献
WO2007/80191 A1, ;
Page/Page column 14-15 ;
WO 2007/080191 A1