2-氰基-N-环丙基-N-[[(2-氟-4-碘苯基)氨基]羰基]乙酰胺合成路线 (共 2 条)
反应条件
sodium hydroxide in water T=80°C; 1 h;
参考文献
JAPAN TOBACCO INC.; SAKAI, Toshiyuki
Patent: WO2005/121142 A1, 2005 ;
Location in patent: Page/Page column 151 ;
反应条件
methanesulfonyl chloride in DMF (N,N-dimethyl-formamide)
T=20°C; 4 h;
参考文献
JAPAN TOBACCO INC.; SAKAI, Toshiyuki
Patent: WO2005/121142 A1, 2005 ;
Location in patent: Page/Page column 150-151 ;