1: HBr / dioxane / 20 h
2: N,N-dimethyl-acetamide / 72 h / Ambient temperature
View Scheme
参考文献
Su, Tsann-Long; Huang, Jai-Tung; Burchenal, Joseph H.; Watanabe, Kyoichi A.; Fox, Jack J.
Journal of Medicinal Chemistry, 1986 , vol. 29, # 5 p. 709 - 715