1: With n-butyllithium in tetrahydrofuran; hexane
T=-78°C; 0.95 h;
2: With boron triethoxide in tetrahydrofuran; hexane
T=20°C; 18 h;
3: With hydrogenchloride in tetrahydrofuran; hexane; water
T=0°C; 0.5 h;
参考文献
BIOLIPOX AB
Patent: WO2005/123673 A1, 2005 ;
Location in patent: Page/Page column 77-78 ;
WO 2005/123673 A1