反应条件
potassium phosphate; palladium 10 on activated carbon; 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl in water; dimethyl sulfoxide T=80°C; 5 h; Inert atmosphere; Product distribution / selectivity;
参考文献
TAKEDA PHARMACEUTICAL COMPANY LIMITED; YAMANO, Mitsuhisa; GOTO, Mitsutaka; KAJIWARA, Takeshi; MAEDA, Hiroyuki; KONISHI, Takahiro; SERA, Misayo; KONDO, Yuichiro; YAMASAKI, Seiji
Patent: WO2012/111849 A1, 2012 ;
Location in patent: Page/Page column 157-158 ;