4-(三氟甲氧基)苄基硼酸频那醇酯合成路线 (共 1 条)
反应条件
1: potassium hydrogen difluoride / methanol; water / 0.5 h / 20 °C
2: boron trifluoride diethyl etherate; copper diacetate / diethyl ether; toluene / 15 h / 20 °C
View Scheme
参考文献
Cazorla, Clement; Metay, Estelle; Lemaire, Marc
Tetrahedron, 2011 , vol. 67, # 45 p. 8615 - 8621