2-氨基-5-甲基-4-(三氟甲基)苯甲酸甲酯合成路线 (共 2 条)
反应条件
cesium fluoride; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in 1,4-dioxane
T=20 - 80°C; 3 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2006/2342 A1, 2006 ;
Location in patent: Page/Page column 56-57 ;
反应条件
pyridine in dichloromethane; toluene
T=0 - 20°C; 2 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2006/2342 A1, 2006 ;
Location in patent: Page/Page column 57-58 ;