2-碘-4-甲基-5-(三氟甲基)苯胺合成路线 (共 2 条)
反应条件
iodine cloride; sodium hydrogencarbonate in methanol; dichloromethane
T=20°C; 3 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2006/2342 A1, 2006 ;
Location in patent: Page/Page column 66 ;
反应条件
pyridine in toluene
T=0 - 20°C; 3 h;
参考文献
ELI LILLY AND COMPANY
Patent: WO2006/2342 A1, 2006 ;
Location in patent: Page/Page column 67 ;