N-(2,6-二氯苯基)乙脒盐酸盐合成路线 (共 1 条)
反应条件
1: 1-amino-2,6-dichlorobenzene With trimethylaluminum in toluene
T=0 - 20°C; 1 h;
2: acetonitrile in toluene
T=80°C; 3 h;
参考文献
EXELIXIS, INC.
Patent: WO2008/73825 A1, 2008 ;
Location in patent: Page/Page column 151 ;
WO 2008/073825 A1