N-[3-(6-氯-吡嗪-2-基)-苯基]-乙酰胺合成路线 (共 1 条)
反应条件
PdCl2[1,3-bis(diphenylphosphino)propane]*CH2Cl2; sodium carbonate in ethylene glycol dimethyl ether
Suzuki coupling; 5 h; Heating;
参考文献
THE WELLCOME TRUST LIMITED
Patent: US2008/15191 A1, 2008 ;
Location in patent: Page/Page column 67 ;