3-甲氧羰基-4-氟苯硼酸合成路线 (共 1 条)
反应条件
1: 2-fluoro-5-iodo-benzoic acid methyl ester With isopropylmagnesium chloride lithium chloride complex in tetrahydrofuran T=-40 - -20°C; 1 h; 2: boron triethoxide in tetrahydrofuran T=-78 - 20°C; 2 h;
参考文献
BIOLIPOX AB; NILSSON, Peter; PELCMAN, Benjamin; KATKEVICS, Martins
Patent: WO2010/103278 A1, 2010 ;
Location in patent: Page/Page column 111 ;