反应条件
1: 97 percent / 1,1,3,3-tetramethylguanidine; BF3*Et2O / acetonitrile / 2.5 h / 25 °C 2: 97 percent / aq. NaOH / ethanol / 3 h / 25 °C View Scheme
参考文献
Gelmi, Maria Luisa; Fontana, Gabriele; Pocar, Donato; Pontremoli, Guido; Pellegrino, Sara; Bombardelli, Ezio; Riva, Antonella; Balduini, Walter; Carloni, Silvia; Cimino, Mauro
Journal of Medicinal Chemistry, 2007 , vol. 50, # 9 p. 2245 - 2248