8-溴-1,6-萘啶-2-甲酰胺合成路线 (共 1 条)
反应条件
1: With 1,1'-carbonyldiimidazole in dichloromethane
6 h;
2: With ammonia in 1,4-dioxane; methanol; dichloromethane
T=20°C; 12 h;
参考文献
Daiichi Sankyo Company, Limited
Patent: EP2380878 A1, 2011 ;
Location in patent: Page/Page column 28 ;