反应条件
1: 2-hydroxy-pyridine With sodium hydride in N,N-dimethyl-formamide
T=0°C; 0.25 h;
2: 4-bromomethyl-fluorobenzene in N,N-dimethyl-formamide
T=0 - 20°C;
参考文献
MERCK and CO., INC.
Patent: WO2006/15159 A2, 2006 ;
Location in patent: Page/Page column 47 ;
WO 2006/015159 A2