反应条件
1: 1.) hexamethyldisilazane, ammonium sulfate, 2.) trimethylsilyl trifluoromethanesulfonate / 1.) reflux, 2 h, 2.) CH2Cl2, RT, 24 h
2: 92 percent / NH3, MeOH / 24 h / 4 °C
View Scheme
参考文献
Mao, David T.; Driscoll, John S.; Marquez, Victor E.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 2 p. 160 - 164
