反应条件
1: 85 percent / potassium carbonate / acetone / 48 h / Heating
2: 1.) acetic acid, iron, 2.) HCl gas / 1.) H2O, 85-95 deg C, 10 h, 2.) ether
3: 95 percent / 20 h / Heating
View Scheme
参考文献
Selassie; Guo; Hansch; Khwaja; Pentecost
Journal of Medicinal Chemistry, 1982 , vol. 25, # 2 p. 157 - 161