4-((3-氨基苯并[e][1,2,4]噻嗪-7-基)氧基)-n-甲基吡啶甲酰胺合成路线 (共 1 条)
反应条件
1: 3-amino-benzo[1,2,4]triazine-7-ol With potassium tert-butylate in N,N-dimethyl-formamide
T=100°C; 0.25 h;
2: 4-chloro-N-methyl-2-pyridinecarboxamide With potassium carbonate in N,N-dimethyl-formamide
T=140°C; 0.5 h;
参考文献
TARGEGEN, INC.
Patent: WO2006/24034 A1, 2006 ;
Location in patent: Page/Page column 30; 66 ;