5-氟-2-(1-哌嗪基)-嘧啶合成路线 (共 2 条)
反应条件
in N-methyl-acetamide; potassium carbonate
参考文献
Neurogen Corporation
Patent: US6284759 B1, 2001 ;
US 6284759 B1
反应条件
in benzene
4 h; Heating; Yield given;
参考文献
Ishizumi; Kojima; Antoku
Chemical and Pharmaceutical Bulletin, 1991 , vol. 39, # 9 p. 2288 - 2300