1: With lithium hexamethyldisilazane in tetrahydrofuran
T=10 - 20°C; 0.166667 h;
2: With hydrogenchloride in tetrahydrofuran; water
T=0°C;
3: With sodium hydroxide in water
pH=14;
参考文献
BOEHRINGER INGELHEIM INTERNATIONAL GMBH
Patent: WO2006/21544 A1, 2006 ;
Location in patent: Page/Page column 64 ;
WO 2006/021544 A1