反应条件
1: 1.) Me2SO4 / 1.) dioxane, THF, 50 deg C, 1 h, 2.) dioxane, THF, H2O, RT, overnight
2: 59 percent / NaN3, NH4Cl / dimethylformamide / 4.5 h / 120 °C
View Scheme
参考文献
Honma; Hanamoto; Hashiyama; et al.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 2 p. 125 - 128
