3-氨基-1-(吡啶-2-基)吡唑合成路线 (共 2 条)
反应条件
potassium tert-butylate in tert-butyl alcohol
T=20°C; 3 h;
参考文献
BANYU PHARMACEUTICAL CO., LTD
Patent: WO2004/37794 A1, 2004 ;
Location in patent: Page 64-65 ;
反应条件
chloranil in chloroform
1 h; Ambient temperature;
参考文献
Doria; Passarotti; Sala; Magrini; Sberze; Tibolla; Buttinoni; Ferrari; Tremolada
Farmaco, Edizione Scientifica, 1985 , vol. 40, # 11 p. 808 - 817