反应条件
hydrogenchloride; sodium hydride 1) THF, reflux, 1 h; 2) H2O, reflux, overnight; Yield given. Multistep reaction;
参考文献
Dukat, M.; Fiedler, W.; Dumas, D.; Damaj, I.; Martin, B. R.; et al.
European Journal of Medicinal Chemistry, 1996 , vol. 31, # 11 p. 875 - 888