反应条件
1: 1.) sodium hydride, 2.) conc. HCl / 1) THF, reflux, 1 h; 2) H2O, reflux, overnight 2: 1.) sodium cyanoborohydride, conc. HCl, 2.) NaBH3CN, NaOAc / 1) H2O, 45 min; 2) pH 6, H2O, 30 min View Scheme
参考文献
Dukat, M.; Fiedler, W.; Dumas, D.; Damaj, I.; Martin, B. R.; et al.
European Journal of Medicinal Chemistry, 1996 , vol. 31, # 11 p. 875 - 888
