反应条件
1.1: caesium carbonate / N,N-dimethyl-formamide
1.2: 1 h / 50 °C
2.1: tetrakis(triphenylphosphine) palladium(0) / N,N-dimethyl-formamide / 0.17 h / 120 °C / Microwave irradiation
View Scheme
参考文献
Brady, Ryan M.; Khakham, Yelena; Lessene, Guillaume; Baell, Jonathan B.
Organic and Biomolecular Chemistry, 2011 , vol. 9, # 3 p. 656 - 658