反应条件
1: 97 percent / ammonium acetate / 24 h / 100 °C 2: 1.) H2, 2.) KOH / 1.) PtO2 / 1.) EtOH, 50 psi, 3 h, 2.) H2O, reflux, 2 h View Scheme
参考文献
Kruse, Lawrence I.; Kaiser, Carl; DeWolf, Walter E.; Finkelstein, Joseph A.; Frazee, James S.; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 2 p. 781 - 789
