N-(5-甲基-6,11-二氧代-6,11-二氢-5H-二苯并[b,e]氮杂卓-10-基)乙酰胺合成路线 (共 2 条)
反应条件
sodium methylate in N-methyl-acetamide; methanol
参考文献
A. Menarini Industrie Farmaceutiche Riunite s.t.l.
Patent: US5080905 A1, 1992 ;
反应条件
Yield given. Multistep reaction. Yields of byproduct given;
参考文献
Perico; Triolo; Viti; Mannucci; Caviglioli; Cocchini; Pestellini; Paoli; Dapporto
Journal of Pharmaceutical Sciences, 1994 , vol. 83, # 2 p. 137 - 142