9-溴-[1,2,4]噻唑[1,5-c]喹唑啉-5(6H)-酮合成路线 (共 1 条)
反应条件
1: in 1-methyl-pyrrolidin-2-one
T=160°C; 1.5 h;
2: With water in 1-methyl-pyrrolidin-2-one
T=25 - 100°C; 0.25 h;
参考文献
Knust, Henner; Stadler, Heinz; Thomas, Andrew William
Patent: US2006/79507 A1, 2006 ;
Location in patent: Page/Page column 18 ;