2-氨基-7-溴-[1,2,4]三唑并[1,5-a]吡啶合成路线 （共 2 条）
反应条件
hydroxylamine hydrochloride; N-ethyl-N,N-diisopropylamine in ethanol T=25°C; 24 h; Reflux; Product distribution / selectivity;
参考文献
F. HOFFMANN-LA ROCHE AG; FLOHR, Alexander; GOBBI, Luca; GROEBKE ZBINDEN, Katrin; KOERNER, Matthias; PETERS, Jens-Uwe
Patent: WO2012/76430 A1, 2012 ;
Location in patent: Page/Page column 90 ;
WO 2012/076430 A1
反应条件
1: 1,4-dioxane / 4 h / 25 °C 2: hydroxylamine hydrochloride; N-ethyl-N,N-diisopropylamine / ethanol / 24 h / 25 °C / Reflux View Scheme
参考文献
US2012/142665 A1, ;
WO2012/76430 A1, ;
WO 2012/076430 A1
