6-溴-吡啶并[2,3-d]嘧啶-2-胺合成路线 (共 1 条)
反应条件
triethylamine in 1-methyl-pyrrolidin-2-one
T=180°C; 0.25 h; Microwave irradiation;
参考文献
BLUEPRINT MEDICINES; BIFULCO, Neil, Jr.; BROOIJMANS, Natasja; HODOUS, Brian, L.; KIM, Joseph, L.; MIDUTURU, Chandrasekhar, V.
Patent: WO2014/11900 A2, 2014 ;
Location in patent: Page/Page column 44; 45 ;