1: With trifluoroacetic acid
T=20°C; 0.5 h;
2: With sodium hydroxide in water
T=0°C;
3: With lithium aluminium tetrahydride in tetrahydrofuran
T=0 - 70°C; 0.5 h;
参考文献
BANYU PHARMACEUTICAL CO., LTD.
Patent: EP1798221 A1, 2007 ;
Location in patent: Page/Page column 28 ;