1-(4-溴苯基)-4-甲基-1H-咪唑合成路线 (共 1 条)
反应条件
copper(l) iodide; trans-N,N-dimethyl-1,2-cyclohexanediamine; caesium carbonate in N,N-dimethyl-formamide
T=110°C; 18 - 20 h;
参考文献
GLAXO GROUP LIMITED
Patent: WO2006/40192 A1, 2006 ;
Location in patent: Page/Page column 40 ;
WO 2006/040192 A1