3-(2,2,2-三氟乙酰基)哌啶-1-羧酸叔丁酯合成路线 (共 1 条)
反应条件
1: With cesium fluoride in tetrahydrofuran
3 h;
2: With hydrogenchloride in tetrahydrofuran; water
1 h;
参考文献
VITAE PHARMACEUTICALS, INC.
Patent: WO2007/117560 A2, 2007 ;
Location in patent: Page/Page column 126 ;
WO 2007/117560 A2