反应条件
sodium hydride
1.) Me2SO, RT, 20 min, 2.) Me2SO, 45-50 deg C, 6 h; Multistep reaction;
参考文献
Awaya, Hiroyoshi; May, Everette L.; Aceto, Mario D.; Merz, Herbert; Rogers, Michael E.; Harris, Louis S.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 4 p. 536 - 539