反应条件
1: 80.3 percent / methanol / 24 h / Ambient temperature
2: 1.) n-BuLi / 1.) ether, hexane, RT, 5 min, 2.) ether, hexane, RT, 36 h
View Scheme
参考文献
Waugh, Kristy M.; Berlin, K. Darrell; Ford, Warren T.; Holt, Elizabeth M.; Carrol, John P.; et al.
Journal of Medicinal Chemistry, 1985 , vol. 28, # 1 p. 116 - 124