反应条件
1: 5-bromo-pyrimidin-2-ylamine With sodium hydride in N,N-dimethyl-formamide
T=0°C; Inert atmosphere;
2: benzyl bromide in N,N-dimethyl-formamide
T=0°C; 2 h; Inert atmosphere;
参考文献
Lu, Jun; Li, Nan-Sheng; Koo, Selene C.; Piccirilli, Joseph A.
Journal of Organic Chemistry, 2009 , vol. 74, # 21 p. 8021 - 8030